Cov tshuaj "Buserelin Ntev" yog ib tug hluavtaws analogue ntawm lub ntuj lawm GnRH. Lub lag luam ntawm qhov cuab tam yog ncaj qha kev sib tw ruaj rau receptors pituitary hlwb thiab tom ntej nraum nce nyob rau hauv cov theem ntawm kev sib deev steroids nyob rau hauv ntshav, uas thaum kawg tau nyob rau hauv tag nrho txhaws ntawm lub thiaj li hu ua gonadotropic pituitary muaj nuj nqi. Raws li ib tug tshwm sim ntawm cov tshuaj "Buserelin Ntev" yog muab ncaj qha suppressing lawm synthesis nyob rau hauv lub gonads, uas manifests nws tus kheej raws li ib tug txo nyob rau hauv testosterone ntau ntau (indices mus post-castration) nyob rau hauv cov txiv neej thiab txo cov ntshav estradiol mus post-menopausal yam ntxwv nyob rau hauv cov poj niam cov neeg mob. Nyob rau hauv thawj cov ntaub ntawv peb yuav hais lus ntawm pharmacological castration, nyob rau hauv lub thib ob - nyob rau hauv postmenopausal los yog ovariectomy.
Cov tshuaj yog tawm nyob rau hauv ib tug lub sij hawm ntawd raws li ib tug lyophilizate yeej tsim los npaj ib tug slurry. Muaj pes tsawg leeg txoj kev npaj no raws li ib tug tub ntxhais lub caij suav txog 4 mg buserelin acetate. Koom haum pab tej yam xwsli carmellose sodium, ib tug copolymer ntawm glycolic thiab dl-lactic acid, polysorbate-80 thiab d-mannitol.
Nrog hais txog kev siv ntawm cov tshuaj, lub koomhaum neeg sawv cev "Buserelin Ntev" rau cov kev kho mob cancer ntawm lub mis thiab hormone-dependent prostate cancer. Nyob rau hauv tas li ntawd, cov tshuaj no yuav siv tau thaum lub sij hawm kev kho mob ntawm endometriosis. Rau cov kev kho mob ntawm uterine fibroids thiab ntxiv lawm tshob (los ntawm IVF cov kev pab cuam) yuav tsum tau pib siv cov tshuaj "Buserelin-Long". Xyuas ntawm cov kws kho mob ua tim khawv txog qhov zoo tau ntawm nws siv rau cov kev kho mob ntawm endometrial hyperplastic dab.
Yog hais tias peb tham txog lub ntsiab contraindications rau kev siv, ces siv cov tshuaj no nruj me ntsis contraindicated rau cov neeg uas muaj ib tug neeg intolerance buserelin acetate, raws li zoo raws li lwm yam ntawm nws txhawb Cheebtsam. Nyob rau hauv tas li ntawd, contraindications muaj xws li cev xeeb tub thiab lactation.
Nyias, nws yuav tsum tau hais tias hais txog cov tau tshwm sim los ntawm kev siv ntawm cov nyiaj "Buserelin-Long", raws li nws yuav ua tau, piv txwv li, qhov ua rau ntawm urticaria, angioneurotic edema thiab hyperemia. Nyob rau hauv tas li ntawd, tej zaum yuav muaj tej yam kev mob xws li demineralization, pw tsaug zog ua cuam tshuam, mob taub hau thiab kev nyuaj siab. Nyob rau hauv poj niam neeg kev mob plab, cov kev hloov nyob rau hauv libido, muaj zog tawm hws, menstrualnopodobnye los ntshav thiab dryness ntawm cov paum mucosa vim kev siv ntawm cov khoom cua tshuaj "Buserelin-Long". Sab los nyob rau hauv cov txiv neej no mas txuam nrog rau exacerbation ntawm lwm tus kab mob, mob txeeb tuav, gynecomastia, thiab "lub raum o." Nyob rau hauv tas li ntawd, nws yuav tsum khij txo nyob rau hauv potency, nce tawm hws, leeg tsis muaj zog nyob rau hauv lub extremities thiab mob pob txha. Ib tug me me muaj pes tsawg tus ntawm cov neeg mob tej zaum yuav muaj kev tshua xws li raws plab mob , thiab pulmonary embolism.