Noj qab haus huv, Npaj
Cov tshuaj "tizanidine": cov lus qhia rau kev siv, synonymous. "Tizanidine-Teva", "tizanidine-Ratiopharm"
Yuav ua li cas noj tshuaj npaum cas kws tshuaj "tizanidine?" Cov lus qhia rau kev siv ntawm lub medicament yog hais hereinafter. Tsis tas li ntawd, los ntawm cov ntaub ntawv ntawm qhov tsab xov xwm koj mam li kawm txog nyob rau hauv dab tsi daim ntawv no yog ua, nws hais tias txhais tau hais tias hais tias ib feem ntawm nws, seb nws muaj kev phiv, thiab contraindications counterparts.
Tus duab, hauj lwm, muaj pes tsawg leeg
Yuav ua li cas yog muaj pes tsawg leeg muaj ib tug yeeb tshuaj "tizanidine?" Cov lus qhia rau Siv hais tias lub active tivthaiv ntawm cov tshuaj no yog tizanidine. Tsis tas li ntawd cov qauv ntawm cov xam tau tias yog medicament muaj raws li cam lactose anhydrous, colloidal silicon dioxide, microcrystalline cellulose thiab stearic acid.
Tshuaj "tizanidine," uas cov kev qhia ntawv yog kos nyob rau hauv lub thawv, ua nyob rau hauv daim ntawv ntawm round dawb cov ntsiav tshuaj. Nyob rau ib sab ntawm lub Paub Faib sawb yog yeeb tshuaj, thiab lub thib ob - labeling lub T4 thiab T2.
pharmacological nta
Yuav ua li cas yog lub mechanism ntawm qhov kev txiav txim "tizanidine" tshuaj? Cov lus qhia rau kev siv ntawd hais tias nws yog ib leeg relaxant. Tom qab tau txais cov ntsiav tshuaj hauv tshuaj active tshuaj thiaj li skeletal leeg tonus, tej lawv tsis kam mus passive suab thiab deceleration ntawm spasmodic tshua thiab li ntawm arbitrary tus nqi.
Los ntawm cov foregoing nws yuav muab tau yooj yim sau hais tias qhov suav hais tias cov tshuaj txhawb nqaij nyhuv relaxing. Qhov no tshwm sim vim cov oppression polisinapticheskie txha caj reflexes. Cov nyhuv no yog vim qhov kev tso tawm ntawm cov amino acids ntawm cov terminals (presynaptic) ntawm tus txha caj interneurons.
pharmacokinetic tsis
Yuav ua li cas yog cov pharmacokinetic tsis muaj tshuaj "tizanidine" (ntsiav tshuaj)? Cov lus qhia rau kev siv nyob rau hauv no hais txog muab tej ntaub ntawv.
Tom qab qhov ncauj thawj coj ntawm lub medicament yog kiag li absorbed. Nws tsis bioavailability yog hais txog 40% (vim nws kim heev thawj pass los ntawm lub siab).
Lub active tshuaj yam khoom uas yog muab faib rau tag nrho cov tshuab thiab ntaub so ntswg. Nws lub koom haum nrog cov nqaijrog ntawm kwv yees li 30%.
Lub ib nrab-lub neej ntawm cov tshuaj yog 2.5 sij hawm. Hais txog 95% ntawm cov tshuaj yog metabolized. Tso tawm kom pom medicament los ntawm ob lub raum (kwv yees li 60%) thiab mob huam (kwv yees li 20%).
indications
Nyob rau hauv tej rooj plaub, muab cov tshuaj "tizanidine?" Kev siv cov tshuaj no yog zoo tshaj plaws nyob rau hauv spastic mob ntawm skeletal leeg, uas tshwm sim thaum neurological kab mob xws li:
- stroke;
- degenerative txha caj qaum kab mob;
- mob myelopathy;
- ntau yam sclerosis.
Tsis tas li ntawd cov tshuaj "tizanidine" qhia nyob pains nyob rau hauv cov nqaij, uas tsim vim lub yeej ntawm cov nqaj qaum.
Contraindications
Lub ntsiab thiab tej zaum qhov tsuas contraindication ntawm cov tshuaj no yog nce neeg mob rhiab heev rau tizanidine. Tsis tas li ntawd, nws yog txwv tsis pub nqa mus siv rau nyob rau hauv nrog xws li "Ciprofloxacin" thiab "Fluvoxamine".
Tshuaj "tizanidine": cov lus qhia rau kev siv
Raws li cov lus qhia, thawj zaug ntau npaum "tizanidine" medicament yog 2 mg.
Txij li thaum cov nyhuv uas cov tshuaj nce mus txog ib tug ncov nyob rau hauv 1-2 xuab moos thiab diluted tom qab 3-6 teev, cov kev kho mob yuav tsum tau nqa tawm ntawm ua mib ntawm 6-8 teev. Yog li, thaum lub sij hawm lub hnub yuav tsum tsis muaj ntau tshaj li 3 lub ntsiav tshuaj.
Cov tshuaj ntawm medicament yog maj nce mus rau 4 mg (ib koob tshuaj). Txawm li cas los, koj ua li ntawd xwb nyob rau hauv rooj plaub yog hais tias, tom qab 4 hnub ntawm kev kho mob cov kev tshwm sim tsis tau qhia.
Tag nrho cov hnub ntau npaum ntawm cov tshuaj yuav tsum tsis txhob muaj ntau tshaj li 36 mg. Nrog kev xav txog ntau npaum units, txais tos ntawm ntau tshaj 16 mg ntawm cov kws tshwj xeeb tau tsis tau kawm.
- Nyob rau hauv lub raum insufficiency. Nrog rau qhov no mob tshuaj kho nrog huab ceev faj.
- Kev txawv txav nyob rau hauv daim siab muaj nuj nqi. Tshuaj "tizanidine" ceev faj yog pom zoo rau cov neeg uas muaj ib daim ntawv uas siab tsis ua hauj lwm. Nyob rau hauv cov neeg mob, tus neeg tshuaj yuav tsum raug txo. Nws yog tsim nyog los lossi xyuas cov theem ntawm aminotransferase. Tus thawj saib xyuas ua ib lub hlis tom qab pib ntawm kev kho mob.
tus neeg mob ntawm overdose
Soj ntsuam cov tsos mob uas tshwm sim tiv thaiv lub keeb kwm ntawm overdose yuav muaj sib txawv kiag li pharmacology. Nyob rau hauv feem ntau tus neeg mob, cov neeg mob muaj nkees, tsis meej pem, kiv taubhau thiab coma. Nyob rau hauv tas li ntawd, cov tshuaj nyob rau hauv high koob tshuaj yuav ua rau tsis ua hauj lwm ntawm cov kev mob plawv, nrog rau cov tshwm sim ntawm bradycardia thiab hypotension.
phiv
Puas muaj tej kev phiv nyob rau hauv cov neeg mob uas tau txais "tizanidine" tshuaj? Cov lus qhia rau kev siv (lus ntawm lub cuab tam yog qhia hereinafter) nyeem tias tus kawm medicament yuav ua rau lub qhov ncauj qhuav, kiv taubhau, hypotension, bradycardia, txo cov ntshav siab, kiv taub hau, mob tu-sauv, qaug zog, tsis muaj zog, qaug zog, yog toog pom, hepatotoxicity, mob ntawm lub siab.
Heev tsis tshua kho nrog cov tshuaj no yeej txhawb cov tsos ntawm Stevens-Johnson syndrome, exfoliative dermatitis, anaphylactic poob siab, ventricular tachycardia, kab mob siab, kev nyuaj siab, qaug dab peg, mob tej pob txha, pob, paraesthesia thiab co.
tshuaj cov kev sib tshuam
Ua ntej siv "tizanidine" tshuaj yuav tsum tau nyeem cov lus qhia kom zoo zoo. Nws qhia txog cov nram qab no nta ntawm nws cov tshuaj cov kev sib tshuam:
- Nyob rau hauv ua ke nrog nrog "ciprofloxacin" thiab "Fluvoxamine" tej zaum yuav ho txo cov ntshav siab, thiab kuj los tsim koj nkees nkees. Nyob rau hauv tas li ntawd, xws complex npaj ua txhaum tib neeg psychomotor zog.
- Tib mus kho mob tshuaj nrog CYP1A2 inhibitors (e.g., "zileuton" "Fluoroquinolones", "Amiodarone", "Mexiletine", "propafenone" "Verapamil," "Cimetidine" "Famotidine" "acyclovir" thiab "ticlopidine") nruj me ntsis txhob.
- Tsis pom zoo ua ke tshuaj "tizanidine" nrog qhov ncauj contraceptives. Yog hais tias tam sim no lub xeev ntawm tus neeg mob yuav tsum tau lub simultaneous thawj coj ntawm cov tshuaj no, cov thawj koob tshuaj yuav tsum tau tsawg heev. Txais tos ntawm siab koob tshuaj ntawm cov tshuaj yuav ua tau kom mob tshwm sim xws li hypotension, bradycardia thiab hypersomnia.
- Muab cov tshuaj no nrog haus dej haus cawv yog tsis pom zoo. Qhov no yog vim lub fact tias cawv tsub kom lub concentration ntawm cov active tshuaj tshuaj nyob rau hauv cov ntshav, thiab qhov no yuav ua rau pliaj teebmeem.
txee lub neej, cia thiab muag khoom tej yam kev mob
Ntsiav tshuaj "tizanidine" dispensed nyob rau hauv pharmacies rau tus kws kho mob tshuaj. Yuav tsum dua li muaj nyob rau ntawm lub chav tsev kub nyob rau hauv ib tug maub qhov chaw. Tsim nyog los tiv thaiv cov tshuaj los ntawm cov me nyuam me.
Txee lub neej ntawm cov nyiaj yog 3 lub xyoo. Tom qab no lub sij hawm nws yog txwv tsis pub noj.
Nqe, txhais thiab analogues ntawm cov tshuaj
Lub sib txawv tshuaj xws li "tizanidine," "tizanidine Ratiopharm" thiab "Teva tizanidine?" Cov lus qhia rau kev siv ntawm cov txhais tau tias muaj tib indications, phiv, contraindications, txoj kev saib xyuas thiab noj tshuaj npaum cas. Qhov txawv tsuas nruab nrab ntawm tus hais cov tshuaj yog lawv manufacturers. Yog li, tag nrho cov ntawm cov nyiaj no yuav muab xam hais tias synonymous.
Raws li rau lub cim "tizanidine" yeeb tshuaj, ces lawv muaj xws li xws cov tshuaj raws li "Sirdalud", "Tizalud" thiab "Sirdalud MP."
Yuav ua li cas npaum li cas yog cov "tizanidine," "tizanidine Teva" thiab "tizanidine Ratiopharm"? Cov kev cai annexed rau cov tshuaj, tsis teb cov lus nug. Yuav kom paub tus nqi ntawm cov txhais tau tias koj yuav tsuas yuav tau mus counter. Raws li ib tug txoj cai, nws yog tsis heev thiab yog hais txog 120-170 Lavxias teb sab rubles (nyob ntawm seb tus xov tooj ntawm tshuaj nyob rau hauv ib lub pob thiab lub chaw tsim tshuaj paus).
Nws yuav tsum tam sim ntawd yuav muab sau tseg tias medicament "tizanidine" muaj ib tug kuj pheej yig tus nqi (piv txwv li, xws analogs li "Sirdalud", "Tizalud" thiab "Sirdalud MR" yog ib tug me ntsis kim, hais txog 240-270 rubles). Uas yog vim li cas feem ntau cov neeg mob muab lawv nyiam mus rau tus thawj yeeb tshuaj.
Tshuaj Xyuas
Tam sim no koj paub yog vim li cas muab tej cov tshuaj raws li "tizanidine," "tizanidine Ratiopharm" thiab "Teva tizanidine." Tus neeg siv kev txaus sab ntawm cov tshuaj mas siv tau raug nthuav saum toj no.
Cov neeg mob uas tau puas tau siv cov tshuaj no, nqa nws nyob rau hauv ntau txoj kev. Feem ntau ntawm cov kev txheeb xyuas kom nws tau los xaus hais tias cov tshuaj "tizanidine" tsis yeej ib txwm ua raws li cov kev cia siab ntawm cov neeg mob.
Muaj coob tus neeg hais tias cov tshuaj no nyob rau hauv ib tug ntawm peb cov neeg mob ua phiv los xws li kev tu-sauv thiab mob ib ce. Zoo ib yam li tshua tshwm sim tam sim ntawd tom qab daim ntawv thov ntawm cov medicament.
Tom qab siv lub ob ntsiav tshuaj, ib co neeg mob xav tias tsis muaj zog, kiv taub hau, thiab kom kuv mus ntuav. Thaum xws li cov tsos mob, kws txawj pom zoo kom tsis txhob tau txais cov nyiaj, los yog lawv siv tej zaum yuav ua rau kom.
Nyob rau hauv tej rooj plaub, tom qab siv "tizanidine" cov neeg muaj teeb meem nrog siab thiab lub plab, thiab lub plawv palpitations.
Nws yuav tsum tau muab sau tseg tias zoo tswv yim los ntawm cov tshuaj nyob rau hauv kev saib xyuas yog tsis yog li ntawd ntau npaum li cas. Ntawm lawv yog cov muaj thiab cov uas tsis muaj nqi ntawm cov tshuaj.
Nyob rau hauv view ntawm lub foregoing nws yuav tsum tau xaus lus tias noj cov tshuaj "tizanidine" thiab nws cov lus ua, tsuas yog yuav tsum tau qhia thiab tsuas yog nyob rau cov tshuaj.
Muab cov loj tus naj npawb ntawm cov nyom tshua, kws txawj tsis pom zoo kom siv cov tshuaj thaum lub sij hawm cev xeeb tub thiab thaum lub sij hawm lub mis noj, txwv tsis pub nws tej zaum yuav detrimental rau lub noj qab haus huv ntawm tus me nyuam los yog me nyuam hauv plab.
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