Noj qab haus huv, Npaj
Efferalgan - cov lus qhia rau kev siv
"Efferalgan" - ib tug nrov antipyretic. Thiab nws muaj pes tsawg leeg yog me ntsis txawv nyob ntawm seb qhov kev tso tawm daim ntawv no. Muaj pes tsawg leeg ntawm lub syrup rau cov me nyuam - paracetamol thiab koom haum pab Cheebtsam: phoov, saccharin, polyethylene glycol, E202, flavors, citric acid, potable dej.
Standard muaj nyob rau hauv lub khob vials ntawm 0,09 litres (ntxiv - ntsuas diav).
Muaj pes tsawg leeg "Efferalgan" (qhov quav): paracetamol, koom haum pab yog cov semi-acylglycerol.
Standard nyob rau hauv cov zauv ntawm 5 tej daim, thiab nyob rau hauv ib lub pob muaj 2 ntim.
Nyob rau hauv nyob tus yeees ntawm effervescent ntsiav tshuaj paracetamol thiab koom haum pab Cheebtsam: qhuav sodium carbonate, povidone, citric acid, saccharin, sorbitol, sodium docusate, ci dej qab zib, E211.
Cov phiaj yog 4 ntsiav tshuaj, thiab tag nrho cov pob - muaj 4, muaj 25 cov ntaub ntawv.
pharmacological los
"Efferalgan" phau ntawv qhia txog cov tshuaj, lub ntsiab active tshuaj yog paracetamol, uas blocks cyclooxygenase-1 thiab 2 tsuas yog nyob rau Cns, yog li exerting cawv rau cov thermoregulatory chaw zov me nyuam thiab kev mob. Nyob rau hauv kub lug ntaub so ntswg qhov kev txiav txim ntawm paracetamol rau COX sim tshwj xeeb, kev peroxidases. Qhov no yog dab tsi piav txog cov yuav luag tiav qhaj ntawv los ntawm anti-inflammatory active tshuaj. Paracetamol yog tsis nyob rau hauv txhua txoj kev muaj feem xyuam rau cov tsim ntawm prostaglandins nyob rau hauv peripheral ntaub so ntswg, uas piav txog nws tag tsis muaj peev xwm los txhawb cov hnyuv mucosa thiab cov ntsha-dej tshuav nyiaj li cas.
Taws tswm ciab "Efferalgan" qhia nthuav txog ob tus neeg saib xyuas muaj analgesic, antiinflammatory thiab antipyretic unexpressed nyhuv.
Paracetamol yog feem ntau nqis kiag li thiab sai sai. Qhov siab tshaj plaws concentration ntawm cov tshuaj yeeb dej caw nyob rau hauv lub ntshiab tshwm sim nyob rau 30-60 feeb. tom qab haus. Sai faib thoob plaws hauv lub cev nqaij, paracetamol yog tsis zoo ua txhua yam rau ntshav cov nqaijrog (mus txog 25%). Nws penetrates rau hauv lub ntshav-hlwb barrier.
Sam metabolism ua los ntawm lub siab. Paracetamol yog tso zis los ntawm lub cev raws li metabolites. Nws yog tso tawm nyob rau hauv cov thawj daim ntawv ntawm tsuas 5% ntawm cov formulation.
zaj lus tim khawv
Tshuaj "Efferalgan" qhia kom cov nram qab no tej yam kev mob thiab cov kab mob:
- ob qho tag nrho antipyretic tshuaj nyob rau hauv cov pa OCR, mob thaum yau pathologies, mob khaub thuas, postprivivochnyh mob, mob thiab inflammatory kab mob uas yog yus muaj los ntawm hyperthermia;
- raws li ib tug analgesic rau ntsis thiab tsis muaj zog mob (mob taub hau, mob nyob rau hauv lub striated nqaij, mob hniav, peripheral paj txhab, kev mob, nyob rau hauv kub nyhiab thiab raug mob).
Contraindications
Contraindications tau txais "Efferalgan" qhia hais xws (tswm ciab, kua syrup)
- loj ua txhaum kev ntawm lub siab los sis mob raum;
- nce nyhav mus rau lub ntsiab tivthaiv;
- kab mob ntawm cov ntshav;
- muaj hnub nyoog ntawm ib lub hlis (rau cov kua syrup) thiab mus txog rau peb lub hlis (rau suppositories 0.08 g);
- tsis muaj tus enzyme G-6-PD;
- los ntshav los yog inflammatory teb nyob rau hauv lub qhov quav (suppository).
Noj ceev faj cov tshuaj yuav tsum tau:
- nyob rau hauv hepatic thiab lub raum tsis ua hauj lwm (ie thaum tsev neeg cholehemia);
- nyob rau hauv lub raum tsis ua hauj lwm yam tsawg kawg nkaus kis ntawm kev siv cov kev npaj nyob rau hauv phoov - 8 teev.
- tsis pom zoo kom siv taws tswm ciab rau raws plab.
Ntsiav tshuaj "Efferalgan" phau ntawv qhia tsis pom zoo kom nyob rau hauv:
- nce nyhav rau lub Cheebtsam;
- tsis tu ncua (nquag) haus cawv;
- Cev xeeb tub (1 thiab 3 trimesters) thiab thaum lub sij hawm noj;
- tsis muaj tus enzyme G-6-PD;
- ua ntej lub hnub nyoog ntawm kaum tsib xyoos (lub cev hnyav - ntawm tsawg tshaj li 50 kg).
Ntsiav tshuaj noj nrog ceev faj:
- mob ntawm daim siab thiab lub raum muaj nuj nqi;
- nyob rau hauv congenital daj ntseg (Dubin-Johnson syndrome, familial cholehemia), kis kab mob siab, hnub nyoog siab tshaj 60 litres, daim siab tus kab mob (cawv) ..
phiv
Sab los thaum noj "Efferalgan" Instruction highlights yog:
- heev tsis tshua muaj - ntuav, xeev siab, kev tsis haum tshuaj (pob, urticaria, pruritus, angioedema);
- cuav along tso quav thiab deurinatsii;
- o ntawm lub qog ua kua week ntawm lub qhov quav;
- heev tsis tshua muaj - thrombocytopenia, anemia, ntshav nyob rau hauv excess ntawm methemoglobin nyob rau hauv cov ntshav tsis muaj peev xwm qe leykotsitopeniya.
Yog hais tias ntev-lub sij hawm kev kho mob nyob rau hauv ntev ntau tej zaum yuav ib nyuag tshuaj lom mus rau lub siab thiab ob lub raum.
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