Noj qab haus huvNpaj

Cov tshuaj "Spitomin": cov lus qhia rau kev siv, indications, contraindications

Niaj hnub no peb qhia rau koj txog cov tshuaj no, raws li "Spitomin". Cov lus qhia rau kev siv, nqe, xyuas, analogs thiab nws cov nta - tag nrho cov sij hawm yog txaus siab cov neeg mob uas tus kws kho mob muaj kws kho cov tshuaj no. Tag nrho cov ntaub ntawv tsim nyog yuav tau pom rau yav tom ntej nyob rau hauv no tsab xov xwm.

Hauj lwm ntawm cov tshuaj, nws zoo lawm, thiab muaj pes tsawg leeg ntawm ntim

Yuav ua li cas yog cov tshuaj "Spitomin"? Cov lus qhia rau kev siv (piav kev npaj muaj yog nyob rau hauv zoo meej) cav hais tias qhov no ntsiav tshuaj dawb ntxhiab, yeej thiab tiaj tus zoo, muaj ib tug chamfer thiab nrog Valium thiab engraving «E151».

Lub cuab tam muaj ib tug buspirone hydrochloride thiab koom haum pab Cheebtsam xws li carboxymethyl starch, lactose monohydrate, magnesium stearate, sodium, microcrystalline cellulose thiab colloidal anhydrous silica.

Nyob rau hauv lub qhov muag ntawm cov tshuaj los nyob rau hauv sawv hlwv packs thiab cartons.

hauv paus ntsiab lus ntawm cov lag luam

Yuav ua li cas nta yog muaj rau cov tshuaj "Spitomin"? Cov lus qhia rau kev siv (ntsiav tshuaj nqi hais hauv qab no) cav hais tias qhov no anxiolytic neeg sawv cev, uas koom mus rau ib tug uas tsis yog-benzodiazepine series thiab muaj ib tug antidepressant nyhuv.

Tsis zoo li lwm yam anxiolytics, cov tshuaj no muaj tsis antiepileptic, sedative, hypnotic thiab myorelaxant zog. Nws paus ntsiab lus ntawm lub lag luam yog ua raws li cov teebmeem ntawm buspirone nyob rau hauv lub dopaminergic thiab serotonergic systems.

Qhov no txhais tau tias xyua thaiv cov hlab qhov dopamine receptors (presynaptic) thiab tsub kom tus nqi ntawm excitation ntawm neurons (dopamine) midbrain.

Yuav ua li cas lwm yam khoom xam qhovkev nyob rau hauv cov tshuaj "Spitomin"? Cov lus qhia rau kev siv hais tias Buspirone yog ib tug xim ib nrab agonist ntawm lub 5-HT1A serotonin receptors. Nws tsis cuam tshuam qhov kev ruaj ntawm benzodiazepine receptors thiab GABA, thiab tsis muaj kev cuam tshuam psychomotor muaj nuj nqi thiab tsis ua rau kam rau ua. Nyob rau hauv tas li ntawd, qhov cuab tam tsis potentiate cov nyhuv ntawm dej cawv haus.

Tus kho nyhuv ntawm qhov suav hais tias cov tshuaj muaj maj thiab tshwm sim tom qab ib los yog ob tom qab kev kho mob.

Kinetics ntawm cov nyiaj

Haum ntawm cov tshuaj "Spitomin", cov lus qhia rau kev siv uas yog qhia hauv qab no, tshwm sim nyob rau hauv lub hnyuv ib ntsuj av. Buspirone yog feem metabolized thaum lub sij hawm cov zaj ntawm lub siab. Nws bioavailability yog 4% thiab lub siab tshaj plaws ntshav concentration yog mus txog tom qab ib teev.

Buspirone yog tso tawm nrog rau cov mis nyuj. Rau cov lus qhia txog lub allergic ntawm cov tshuaj los ntawm lub placental barrier tsis.

Kev npaj muab los ntawm faeces rau tsib lub sij hawm.

zaj lus tim khawv

Los ntawm dab tsi yog tshuaj "Spitomin" ntsiav tshuaj? Cov lus qhia rau kev siv qhia cov nram qab no indications:

  • autonomic kawg syndrome;
  • ntxhov siab vim teeb meem yog generalized;
  • ntsoos ntsoos syndrome haus cawv (raws li adjuvant therapy);
  • panic teeb meem ;
  • depressive ntshawv siab (raws li adjuvant therapy).

Contraindications

Nyob rau hauv tej rooj plaub, nws yog tsis pom zoo kom siv tshuaj "Spitomin"? Cov lus qhia rau kev siv hais tias cov nram qab no pathologies thiab tej yam kev mob nyob rau hauv uas lub koob tshuaj yog ua rau:

  • glaucoma;
  • npau taws me ntsis rau cov khoom xyaw tshuaj;
  • myasthenia Heavy kev;
  • raum insufficiency, mob;
  • me muaj hnub nyoog;
  • simultaneous txais tos ntawm Mao inhibitors ;
  • lactation;
  • thaum lub sij hawm cev xeeb tub.

Nrog kho mob yog muab nyob rau hauv daim siab mob npuas paug thiab lub raum tsis ua hauj lwm.

Medicament "Spitomin": cov lus qhia rau kev siv

Analogs ntawm cov tshuaj yuav tsum tau muab nthuav hauv qab no.

Ntawm cov nyiaj yuav tsum tau noj nyob rau hauv tib lub sij hawm ntawm lub hnub, ua ntej los yog tom qab ib tug noj mov.

Cov tshuaj no yog txwv tsis pub siv puav (xav tau) rau cov kev kho mob ntawm kev ntxhov siab vim, txij li thaum nws kho nyhuv muaj tsuas yog tom qab rov siv.

Cov tshuaj ntawm cov tshuaj no yog xaiv ib lub zuj zus. Feem ntau, nws yog 15 mg. Nws yuav tsum tau muab faib ua 2-3 koob tshuaj.

Qhov siab tshaj plaws ib koob tshuaj yog 30 mg thiab lub siab tshaj plaws txhua hnub - 60 mg.

Nyob rau hauv cov neeg laus kho ntawm koob tshuaj yog yuav tsum tau. Thaum lub raum los yog hepatic medicament yuav tsum tau siv nrog ceev faj nyob rau hauv me me koob tshuaj.

phiv

Feem ntau cov tshuaj "Spitomin" zoo taus. Tsuas yog nyob rau hauv tej rooj plaub, qhov cuab tam yog tej yam ua txhaum cai:

  • mob hauv siab, teeb meem tsaug zog, tsaus muag, kiv taub hau, hypotension, mob taub hau, tawg;
  • tshee ntxhov siab vim, cerebral lub plawv mob, dysphoric tshua, decompensation ntawm lub plawv tsis ua hauj lwm, muaj rhiab heev rau suab nrov, heart attack myocardial infarction, dysphoria, cardiomyopathy, suicidal xav, bradycardia;
  • depersonalization, txias intolerance, zoo siab, claustrophobia, hyperkinesis, tinnitus, ntxhov siab vim, khaus nyob rau hauv lub qhov muag, nkees, lub qhov muag liab liab, hallucinations, thob-quav, tsis meej pem, psychotic mob;
  • qhov muag plooj tsis pom kev, laryngitis, conjunctivitis, o ntawm lub qhov ntswg mucosa, impaired saj, ib tug zoo nkaus li heaviness nyob rau hauv lub hauv siab, inner pob ntseg mob, hyperventilation, qhov muag mob, tsis muaj cua, photophobia, epistaxis, nce intraocular siab;
  • galaktoreyu, xeev siab, thyroid kev puas tsuaj, flatulence, nocturnal enuresis, anorexia, qab los noj mov nce, dysuria, salivation, coj khaub mob, plab hnyuv los ntshav, ncua ejaculation thiab lwm yam.

Nqe, analogues, xyuas

Tus nqi ntawm no neeg sawv cev yog hais txog 600 rubles. Yog hais tias yuav tsum tau, nws yog hloov nrog ib tug analog xws li "Buspirone Sandoz."

Consumer xyuas qhia tias cov tshuaj nyob rau hauv lo lus nug yog ib tug zoo anxiolytic neeg sawv cev. Txawm li cas los, nws yuav noj xwb ib tug kws on lub hom phiaj rau ib tug ntev lub sij hawm (tsis puav).

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